Биологическая активность
Bupropion, also known as amfebutamone and BW 323, is a norepinephrine–dopamine reuptake ингибитор (NDRI) and a nicotinic рецептор антагонист. However, its effects on dopamine are weak and clinical significance is contentious. Chemically, bupropion is an aminoketone that belongs to the class of substituted cathinones and more generally that of substituted amphetamines and substituted phenethylamines.
Оригинал на английском
Bupropion, also known as amfebutamone and BW 323, is a norepinephrine–dopamine reuptake inhibitor (NDRI) and a nicotinic receptor antagonist. However, its effects on dopamine are weak and clinical significance is contentious. Chemically, bupropion is an aminoketone that belongs to the class of substituted cathinones and more generally that of substituted amphetamines and substituted phenethylamines.
Химические свойства
- CAS №
- 31677-93-7
- Брутто-формула
- C₁₃H₁₉Cl₂NO
- Мол. масса
- 276.20 г/моль
- Синонимы
- Bupropion, Wellbutrin, Zyban; BW 323; BW-323; BW323. NSC 315851.
Хранение и физические свойства
- Условия хранения
- 2 года -20°C порошок, 2 недели 4°C в ДМСО, 6 мес. -80°C в ДМСО
Безопасность и документация
Только для научно-исследовательского применения. Не предназначено для использования у пациентов или в качестве лекарственного средства.