Биологическая активность
Darodipine, also known as PY-108068, is a мощный a calcium антагонист. Darodipine dose-depentently blocks I(Ca,L) in rat isolated cardiomyocytes. Darodipine exerts protective effects against free-radical-induced electrophysiological alterations independently of its calcium antagonistic properties; this effect is possibly due to trapping of specific radical species. .
Оригинал на английском
Darodipine, also known as PY-108068, is a potent a calcium antagonist. Darodipine dose-depentently blocks I(Ca,L) in rat isolated cardiomyocytes. Darodipine exerts protective effects against free-radical-induced electrophysiological alterations independently of its calcium antagonistic properties; this effect is possibly due to trapping of specific radical species. .
Химические свойства
- CAS №
- 72803-02-2
- Брутто-формула
- C₁₉H₂₁N₃O₅
- Мол. масса
- 371.39 г/моль
- SMILES
- O=C(C1=C(C)NC(C)=C(C(OCC)=O)C1C2=CC=CC3=NON=C23)OCC
- Синонимы
- PY-108068; PY108068; PY108068; PY108-068; PY-108-068 и ещё 2
3D-структура молекулы
Вращайте мышью · Колесо — масштаб
Безопасность и документация
Только для научно-исследовательского применения. Не предназначено для использования у пациентов или в качестве лекарственного средства.