JNJ-31020028 is a селективный brain penetrant антагонист of neuropeptide Y2 рецептор with high affinity(pIC50=8.07, human; pIC50=8.22 rat); >100-fold селективный versus human Y1/Y4/Y5 receptors.
Оригинал на английском
JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22 rat); >100-fold selective versus human Y1/Y4/Y5 receptors.