Биологическая активность
Ethacizine hydrochloride (Ethacizin; NIK-244) is a Class Ic antiarrhythmic agent, which means it is part of a group of drugs that primarily act by blocking sodium channels in the heart. This class of antiarrhythmic agents is known for their мощный effects on slowing conduction in the heart, particularly in the atria, ventricles, and the His-Purkinje system.
Оригинал на английском
Ethacizine hydrochloride (Ethacizin; NIK-244) is a Class Ic antiarrhythmic agent, which means it is part of a group of drugs that primarily act by blocking sodium channels in the heart. This class of antiarrhythmic agents is known for their potent effects on slowing conduction in the heart, particularly in the atria, ventricles, and the His-Purkinje system.
Химические свойства
- CAS №
- 57530-40-2
- Брутто-формула
- C₂₂H₂₇N₃O₃S.HCl
- Мол. масса
- 449.99 г/моль
- SMILES
- Cl.CCOC(NC1C=CC2=C(N(C3=CC=CC=C3S2)C(CCN(CC)CC)=O)C=1)=O
- Синонимы
- Carbamic acid,[10-[3-(diethylamino)-1-oxopropyl]-10H-phenothiazin-2-yl]-, ethyl ester,monohydrochloride (9CI); ETHACIZINE HCL; ethyl N-[10-(3-diethylaminopropanoyl)phenothiazin-2-yl]carbamate hydrochloride; ethyl N-[10-[3-(diethylamino)propanoyl]phenothiazin-2-yl]carbamate,hydrochloride; Ethacizine hydrochloride
3D-структура молекулы
Вращайте мышью · Колесо — масштаб
Хранение и физические свойства
- Условия хранения
- 2 года -20°C порошок, 2 недели 4°C в ДМСО, 6 мес. -80°C в ДМСО
Безопасность и документация
Только для научно-исследовательского применения. Не предназначено для использования у пациентов или в качестве лекарственного средства.